Skip to content
Research Monograph

AOD-9604 (Anti-Obesity Drug 9604)

Also Known AsAOD 9604 · Tyr-hGH Fragment 177-191 · hGH Fragment

Molecular Weight1815.08 g/mol
Discovered1998
Citations3 peer-reviewed
Research Areas3 domains
Background

Developed by Frank Ng and colleagues at Monash University, Melbourne, Australia as a modified fragment of human growth hormone (amino acids 177-191). The fragment was identified as the lipolytic region of hGH, with the addition of a tyrosine residue at the N-terminus improving stability and receptor binding without stimulating IGF-1 or exhibiting growth-promoting effects.

Mechanisms of Action

How AOD-9604 Works

01

Beta-3 Adrenergic Receptor Pathway

AOD-9604 mimics the lipolytic mechanism of hGH by stimulating beta-3 adrenergic receptors in adipose tissue, triggering hormone-sensitive lipase (HSL) activation and subsequent triglyceride hydrolysis. Unlike full hGH, it does not activate the JAK2/STAT5 growth pathway.

β3-adrenergic receptorhormone-sensitive lipaseadipocytes
02

Anti-Lipogenic Activity

Inhibits lipogenesis (fat formation) by suppressing key lipogenic enzymes including fatty acid synthase and acetyl-CoA carboxylase. This dual action (promoting fat breakdown while preventing fat formation) distinguishes it from compounds that only affect one side of the equation.

fatty acid synthaseacetyl-CoA carboxylaselipogenic pathway
03

Cartilage Regeneration

Emerging research demonstrates chondroprotective and regenerative effects. AOD-9604 stimulates proteoglycan and collagen synthesis in cartilage tissue, promoting extracellular matrix production in osteoarthritic joints.

chondrocytesproteoglycanscollagen type II
Evidence-Graded Research Areas

Published Research

Strong
Moderate
Emerging
Preclinical

Obesity & Fat Metabolism

Moderate

Phase 2 clinical trials demonstrated dose-dependent weight loss over 12 weeks in obese subjects without affecting IGF-1 levels or causing diabetogenic effects. Animal studies consistently show reduction in body fat without affecting lean mass. AOD-9604 received GRAS (Generally Recognized As Safe) status from the US FDA in 2014.

Osteoarthritis & Cartilage Repair

Moderate

Preclinical studies demonstrate stimulation of cartilage repair via enhanced proteoglycan synthesis. A proprietary formulation (i-Body) has completed Phase 2 clinical trials for knee osteoarthritis showing improved pain scores and function. Mechanism is distinct from its metabolic effects.

Growth Hormone Dissociation

Strong

AOD-9604 is a key research tool for understanding which domains of human growth hormone are responsible for different biological effects. It demonstrates that the lipolytic, anti-lipogenic, and chondroprotective actions of hGH can be isolated from its growth-promoting and diabetogenic effects.

Safety Profile

AOD-9604 received GRAS (Generally Recognized As Safe) status from the US FDA in 2014 for use as a food ingredient. Phase 2 clinical trials reported no significant adverse effects versus placebo. Key safety advantage: does not affect IGF-1, glucose homeostasis, or growth parameters, eliminating the metabolic risks associated with full hGH.

Handling & Storage

Reconstitute with bacteriostatic water. AOD-9604 is a stable peptide fragment with good aqueous solubility. Store reconstituted solution at 2-8°C. Lyophilized powder stable at -20°C for 24+ months.

References & Citations

Peer-Reviewed Literature

  1. 1

    Increase of fat oxidation and weight loss in obese mice by chronic treatment with human growth hormone or a modified C-terminal fragment

    Heffernan MA, Thorburn AW, Fam B, et al.

    International Journal of Obesity, 2001PubMed 11753577DOI
  2. 2

    Metabolic studies of a synthetic lipolytic domain (AOD9604) of human growth hormone

    Ng FM, Sun J, Sharma L, et al.

    Hormone Research, 2000PubMed 11146374DOI
  3. 3

    Safety and tolerability of the hexadecapeptide AOD9604 in humans

    Stier H, Vos E, Kenley D.

    Journal of Endocrinology and Metabolism, 2013
Frequently Asked Questions

AOD-9604 FAQ

What is AOD-9604?

AOD-9604 (Anti-Obesity Drug 9604) is a modified fragment of human growth hormone consisting of amino acids 177-191 with an additional N-terminal tyrosine. It was designed to retain the fat-metabolizing properties of growth hormone while eliminating its growth-promoting and diabetogenic effects. It received FDA GRAS status in 2014.

How is AOD-9604 different from HGH?

AOD-9604 is a small fragment (16 amino acids) of the full 191-amino-acid hGH molecule. It retains the lipolytic (fat-burning) and anti-lipogenic (fat-formation-preventing) activities but does NOT stimulate IGF-1, does not promote growth, and does not cause insulin resistance — eliminating the major safety concerns of full growth hormone.

Does AOD-9604 have FDA status?

Yes. In 2014, AOD-9604 received GRAS (Generally Recognized As Safe) status from the US FDA for use as a food ingredient. This is not a drug approval but confirms safety for human consumption at food-grade levels. Research-grade AOD-9604 is sold for investigational use only.

Available for Research

AOD-9604 Products

All compounds 99%+ purity, verified by Janoshik Analytical. GMP-manufactured lyophilized powder.

Buy 3, Save 30%
AOD
Lyophilized Powder
99%

The fat-burning fragment of growth hormone — targets and destroys stubborn body fat (especially belly fat) without touching muscle, blood sugar, or hormone levels.

  • Burns fat without affecting blood sugar or growth hormone levels
  • Targets stubborn belly fat specifically
$52.79
Related Compounds

Explore Related Research

Buy 3, Save 30%bestseller
Sem
Lyophilized Powder
99%

The weight loss revolution — the same molecule in Ozempic that helps millions lose 15-20% of body weight by silencing food cravings and resetting appetite at the brain level.

  • Lose 15-20% of body weight without willpower or starvation
  • Completely eliminates food noise and constant cravings
$98.99
Buy 3, Save 30%trending
5-A
Oral Capsules
99%

5-Amino-1MQ

50mg × 60 Capsules

Burns fat at the cellular level — blocks the enzyme that makes fat cells expand, shrinking them while you keep eating normally.

  • Shrinks fat cells without changing your diet
  • Blocks the enzyme (NNMT) that makes fat cells grow
$209.99
Buy 3, Save 30%trending
MOT
Lyophilized Powder
99%

MOTS-c

10mg

Exercise in a molecule — activates your metabolism, burns fat without dieting, and gives your cells the energy boost of a hard workout.

  • Burns fat by activating your body's metabolic furnace (AMPK)
  • Mimics the benefits of exercise at the cellular level
$99.99

Disclaimer: This monograph is provided for educational and research purposes only. G26x Peptides products are sold exclusively as research chemicals. They are not intended for human consumption, therapeutic use, or as dietary supplements. All research should be conducted in compliance with applicable laws and institutional review board protocols. Information presented here is sourced from published peer-reviewed literature and does not constitute medical advice.